苯酰胺

After the use niter benzene even treatment and the treatment all around, separately makes the electroencephalogram inspection to two groups of case of illness.results: after the use niter benzene even treatment all around, the treatment group electroencephalogram restores quickly to the comparison group, exceptionally leads obviously to be lower than the comparison group.conclusions: the niter benzene is even is treats the recovery period fluorine acetamide to be poisoned patient's effective method, may enable his/her the brain harm to obtain the as soon as possible repair, improves the brain function, makes the unusual electroencephalogram to restore normal or the change for the better as soon as possible.

在使用硝苯地平治疗前和治疗4周后，分别对两组病例均作脑电图检查。结果：使用硝苯地平治疗4周后，治疗组脑电图恢复快于对照组，异常率明显低于对照组。结论：硝苯地平是治疗恢复期氟乙酰胺中毒患者的有效手段，可使其脑损害得到尽快修复，改善脑功能，使异常的脑电图尽早恢复正常或好转。

Benzyloxy benzoyldimethylsulfoxide was prepared by the reaction of ethyl 4-benzyloxybenzoate and dimethyl sulfoxide in the presence of sodium hydride, followed by Pummerer reaction with concentrated hydrochloric acid to afford eo-hydroxy-co-thio-methyl-(4/-benzyloxy) acetophenone, which reacted with urea, thiosemicarbazide, semicarbazide hydrochloride and o-phenylenediamine to give imidazolidine-2,4-dione, l,2,4-triazine-3- one and quinoxaline derivatives, respectively.

本文用4-苄氧基苯甲酸乙酯和二甲亚砜为原料，在氢化钠存在下反应，合成了(4′-苄氧基)-苯甲酰基-二甲亚砜。研究了该亚砜在浓盐酸的存在下发生的Pummerer重排反应，用重排产物ω-羟基-ω-甲硫基-(4′-苄氧基)-苯乙酮分别与尿素、氨基脲、氨基硫脲和邻苯二胺反应合成了2，4-咪唑啉-二酮、1，2，4-三嗪-3-酮、喹喔啉等含氮杂环化合物。

The paper proposed a possible binding mode of MS-275, a benzamide histone deacetylase inhibitor, to HDAC by intensive docking study.

通过计算机模拟的对接过程研究，发现了MS-275--一种苯甲酰胺类的组蛋白去乙酰酶抑制剂与酶的可能的全新结合方式。

A series of 2-acetylformanilides were prepared,followed by thiolation with Lowesson reagent to afford 2-acetylthioformanilides,which further reacted with Mn3·2H2O in glacial acetic acid under microwave irradiation to afford 2-acetyl benzothiazole s.

合成了一系列的硫代酰胺，研究了它们在微波辐射醋酸锰作用下发生氧化自由基环化反应，成功地合成了一系列2-乙酰基苯并噻唑衍生物，其结构经红外光谱、核磁共振谱和质谱得到了证实

The synthesis of poly{2-4-[bi(4-tetrabutylphenylamino]phenylphenylenenvinylene} was beginwith 4-tetrabutylbenzoic,through acylation、Hoffmann rearrangement、bromization、idionization、Ullmann reaction、bromization、condensepolymerization.

聚{2-[4-二(4-叔丁基苯胺基苯基]苯撑乙烯}是以对叔丁基苯甲酸为原料，经酰氯化、酰胺化、Hoffmann降解、碘化、Ullmann反应、溴化、缩聚反应得到。

In this analogue, the hydrogen of amide group could still form a hydrogen bond with the oxygen of ester bond and the ester bond was isosteric with peptide bond.

我们合成了甜味肽的类似物L-天冬酰氨酰-L-α-羟基苯丙酸甲酯，将甜味肽的天冬氨酸替换为天冬酰胺，肽键替换为酯键。

A series of new DB21C7 derivatives with straight arm chains (crown 1 ~ 20) were firstly synthesized, and a thorough and systematic study about the influence of side arms which containing different length polymethylene and certain functional groups on extraction capacity of the parent DB21C7 was made.

本文利用DB21C7中苯环的活性，通过苯环上的亲电取代反应，首次设计合成了二苯并-21-冠-7桥连的二酮、直链烷烃、二醇、二酮酸、二烷酸以及二酰胺，共20个DB21C7取代衍生物，并以IR、~1H NMR、MS和元素分析进行了表征。

Based on 26B4APBN monomer, polyamic acid was obtained by polymerization with pyromellitic dianhydride, and further imidized into polyimide film by heating process.

由二胺单体和均苯四甲酸二酐进行聚合得到26B4APBN/PMDA聚酰胺酸，再经热亚胺化得到聚酰亚胺薄膜；测试了该薄膜的接触角，讨论了单体分子结构对聚合物接触角的影响。

Methods 2-(piperazin-1-yl)-1-(pyrrolidin-1-yl)ethanone (2) was synthesized from pyrrolidine via amidation and substitution, followed by treating with chloroacetyl chloride and triphenylphosphine in a "one pot" manner to give the corresponding phosphonium chloride 3 in a stable and pure form after crystallization from isopropanol.

以四氢吡咯为原料，先与氯乙酰氯成酰胺，再与哌嗪发生取代反应制得中间体［（1-四氢吡咯基）甲基］哌嗪(2)；化合物2与氯乙酰氯和三苯基膦反应，经异丙醇重结晶得到稳定的有机鏻盐(3)；化合物3与3，4，5-三甲氧基苯甲醛发生Wittig反应，再与马来酸成盐得目标化合物马来酸桂哌齐特(1)。

Bezaldehyde was used as protective agent in first method.S-Epichloeohydrin was aminated and acidulated to give(2S)-1-Amino-3-chloro-propanol Salts.The acetylation of (2S)-1-Amino-3-chloro-propanol by acetic anhydride produced the intermediate-N-[2--3-chloropropyl]acetamide.And then at 20℃,in the presence of lithium tert-butoxide,benzyl 3-fluoro-4-morpholinophenyl carbamate react with-N-[2--3-chloropropyl]acetamide to give linezolid in total yield of 43.6%.

路线一采用苯甲醛作保护剂，使S-环氧氯丙烷氨解、酸化生成S-1-氨基-3-氯-2-丙醇盐酸盐，然后经乙酰化反应后，生成中间体-N-[2-乙酰氧基-3-氯丙基]乙酰胺，再用N-(3-氟-4-吗啉苯基)氨基甲酸苄酯和中间体在催化剂叔丁醇锂存在下25℃反应生成利奈唑酮，总产率达到43.6%。

The split between the two groups can hardly be papered over.

这两个团体间的分歧难以掩饰。

This approach not only encourages a greater number of responses, but minimizes the likelihood of stale groupthink.

这种做法不仅鼓励了更多的反应，而且减少跟风的可能性。