氧化合物

Results Compound albicanyl caffeate displayed strong antifungal property with MIC 4 μg/ml, while moderate antifungal effects (MIC16 μg/ml)were observed with compounds emodin, resveratrol, 3,4'-difluorostilbene, 2,2'-difluorostilbene and 2,3',5'-trifluorostilbene. Pakyonol, catechin, ampelopsin A, 3,4,4'-trihydroxyl- bibenzyl, 2,4'-difluorostilbene, 4-fluorostilbene,2-methyloxy-4'-fluorostilbene showed lower activity with MIC 32 μ g/ml.

结果化合物albicanyl caffeate对白色念珠菌表现出强的抗真菌活性，MIC为4μg/ml；而化合物大黄素、白藜芦醇、3，4'-二氟二苯乙烯、2，2'-二氟二苯乙烯及2，3'，5'-三氟二苯乙烯显示出中等程度的抗真菌活性，MIC为16μg/ml；双联苄pakyonol、多酚类儿茶素、白藜芦醇二聚体野葡萄素A、3，4，4'-三羟基联苄、2，4'-二氟二苯乙烯、4-氟二苯乙烯及2-甲氧基-4'-氟二苯乙烯显示出较弱的抗真菌活性，MIC为32 μg/ml。

Aim To design and synthesize a series of 2--(4-cyclopentyloxy-3-methylbenzylidene)cyclopentanone arylamine Mannich bases,and to determine their antitumor activities in vitro.

目的设计合成一系列2--(4-环戊氧基-3-甲氧基苯亚甲基)环戊酮Mannich碱类化合物，并对其抗肿瘤活性进行体外试验。

A novel liquid crystalline compound named p-phenylenediamine di 4-[2- benzamide] was synthesized from allyl 2-hydroxyethylether, ethyl 4-hydroxybenzoate and p-phenylenediamine.

以乙二醇单烯丙基醚、对羟基苯甲酸乙酯、对苯二胺为原料合成了末端为不饱和双键的芳香聚酰胺溶致型液晶化合物——二对烯丙氧基乙氧基苯甲酰对苯二胺，最佳合成的摩尔比为∶羧酸∶对苯二胺∶吡啶=2。

The pyrimidine lead compound is obtained via herbicidal activity screen. The optimization of lead compound leads to find the good pyrimidine benzylamine candidates with highly effective herbicidal activity. The novel herbicidal mechanism of pyrimidine benzylamine is put forward. N-(2-bromophenyl)-2-(4, 6-dimethoxypyrimidin-2-yloxy)benzylamine (103-1) has potential as a new selective post-emergent herbicide in oilseed rape.

通过系统的研究工作，发现了具有除草活性的嘧啶先导结构，经结构优化，筛选出具有高除草活性的嘧啶苄胺类优选结构，发现并提出了此类化合物的除草作用新机理，最终经田间试验证实了N-(2-溴苯基)-2-(4，6-二甲氧基-2-嘧啶氧基)苄胺(103-1)可作为超高效油菜田除草剂进行工业性的研究与开发。

Direct competitions of intramolecular C - H insertions into benzylic C - H and 4-nitroor 4-methoxy substituted benzylic C - H of methyl 2-diazo-3-oxo-6-(4-substituted phenyl)-4-(2-phenylethyl)hexanoate 44a and 44b catalyzed by Rh-mediated carbenoid were alsoinvestigated, and the relative reactivities obtained by compound 44a or 44b were comparableto those obtained by indirect method.

此外，还研究了Rh催化分解下，对位硝基取代或甲氧基取代的4-(2-苯基乙基)-6-(4-取代苯基)-2-重氮基-3-氧代己酸甲酯44a、44b苯甲位C-H插入反应的相对速率，与化合物47a和47f得到的结果比较，数据平行。

In this paper, two novel Organic- Inorganic Hybrid Compounds Containing POMs were achieved by selecting POMs with unique structure and properties and organic ligands with bipyridyl groups as building blocks and transition mental cation as templating through hydrothermal reaction.

本课题选择结构和性能独特的多金属氧酸根和多齿有机配体作为构件，以金属离子作为模板合成出新型多金属氧酸盐无机－有机杂化化合物。

He first synthesis of the precursor 45b of Tuxpanolide was accomplished fromβ-alkoxy aldehyde and β-acetoxy-γ-butyrolactone by the Aldol reaction.

uxpanolide的合成前体45b的首次不对称合成：以β-烷氧基开链醛和β-乙酰氧基-γ-丁内酯参与的Aldol醛醇缩合反应首次得到了前体化合物45b。

In this dissertation, I will represent my studies on the nitration of Chalcone derivatives, reaction of epoxide ketone, and the aromatization of 3,5-disubstitued 2-isoxazolines with nitric oxide.

本文主要研究了：(1)NO与查尔酮及其衍生物的硝化反应，反应以较高的产率得到了a-硝基化合物；(2)NO对环氧酮的开环反应，反应生成了顺式羟基硝酸酯；(3)3，5-二取代的-2-异恶唑啉在NO作用下可以发生芳环化反应，生成了对应的2-异恶唑化合物。

The method comprises: utilizing arctiin as the precursor compound, and converting arctiin into 4, 4'-dihydroxy enterolactone by intestinal bacteria in an anaerobic condition. 4, 4'-dihydroxy enterolactone is lignin compound, and can be converted into phytoestrogen in human intestinal canals.

本发明是以牛蒡苷为先导化合物，在厌氧条件下，以肠道细菌将牛蒡苷转化为4，4′-二羟基肠内酯。4，4′-二羟基肠内酯为木脂素类化合物，在人的肠道中能被转化为植物雌激素―肠内酯而发挥药理作用。

By bioactivity-guided isolation, 14 compounds were obtained from the active fractions. 13 of them were determined as 9,9'-dihydroxy-8,8'-dimethoxy- l,r-methyl-lH,lH'-[4,4']binaphtha

本研究利用稻瘟霉筛选体系对红葱的60％乙醇提取物及其氯仿、正丁醇和水的萃取部分进行了活性筛选，并对活性部位的活性化学成分进行了跟踪分离，从中分离得到十四个化合物，利用物理化学和光谱学的方法对其中十三个化合物的结构进行了鉴定，分别为9，9'-二羟基-8，8'-二甲氧基-1，1'-二甲基-1H，1H'-[4，4']双萘并

She gently rebuff ed him, but agreed that they could be friends

她婉言拒绝了，但同意作为朋友相处。

If in the penal farm, you were sure to be criticized.

要是在劳改农场，你等着挨绳子吧！