抑制的

GnRH could markedly suppress progesterone secretion of cultured GCs with or without FSH and LH co-treatments. E〓 could invert the suppression of GnRH completely, also had the additive action on secreting progesterone with GnRH co-treatment. Mel partially released the suppression action of GnRH.

GnRH能强烈地抑制体外培养的颗粒细胞分泌孕酮，其抑制作用几乎不受FSH和LH影响；Mel仅表现部分地缓解了GnRH的抑制效应，但没有逆转。E〓不仅可以完全逆转GnRH的抑制作用，进而与GnRH叠加促进颗粒细胞分泌孕酮。

They were reversible un-competitive inhibitors, and their inhibition constants of free enzymeK(subscript I were 254.00 and 136.78 mmolL^(-1), respectively. Urea was reversible mixed-type inhibitor, and its inhibition constants of free enzymeK(subscript I and enzyme-substrate complexK(subscript IS were determined to be 379.02 and 1182.00 mmolL^(-1), respectively.

Na2SO3和H2O2对酶的抑制均表现为可逆反竞争性类型，它们对游离酶的抑制常数K(下标 I分别为254.00和136.78 mmolL^(-1)；尿素对酶的抑制表现为可逆的混合型抑制，它对游离酶的K和对酶－底物复合物的抑制常数K(下标 IS分别为379.02和1182.00 mmolL^(-1)。

Analysing ustiloxins inhibiting plant cell mitosis The inhibition experiment of growth of garlic radicle showed that there were more cells in the telophase stage in the garlic radicle dealed with culture filtrate of Ustilaginodea virens than those dealed with H2O. The cell volume of the former was bigger than that of the latter. So it seemed that ustiloxins could inhibit the cell mitosis, but not in the cell elongation.

毒素对植物细胞分裂的抑制作用分析：用大蒜根尖做抑制试验，发现用稻曲病菌培养滤液处理过的大蒜根尖呈分裂末期的细胞数目明显多于相同条件浙江大学硕士学位论文下对照的数目，抑制率为69%，且细胞明显比对照的细胞大，说明毒素抑制根尖细胞的有丝分裂，但不能抑制细胞的伸长。

objective effects of plant tannins,chebulinic acid and tellimagrandin i on chemically induced hemoglobin synthesis in k562 cells were investigated.methods the hemoglobin synthesis situation was assayed with benzidine staining.erythroid antigens glycophorin a expression on the surface of k562 cells was labeled by direct immunofluorescence using fluorescein isothiocyanate-conjugated anti-gpa antibodies.then flow cytometric analysis was performed to detect gpa expression levels on surface of the cells.results both chebulinic acid and tellimagrandin i could inhibit the hemoglobin synthesis of butyric acid and hemin-treated k562 cells in a concentration-dependant manner.however,the ba-induced k562 cells were more sensitive to two tannins than heroin-induced cells.conclusion chebulinic acid and tellimagrandin i have inhibitory effect on the erythroid differentiation.

目的 研究可水解单宁诃子酸和特里马素i对氯化高铁血红素和丁酸钠诱导k562细胞红系分化的影响。方法四甲基偶氮噻唑蓝法分析诃子酸和特里马素i对k562细胞生长的影响，联苯胺染色法检测血红蛋白合成情况，应用免疫荧光和流式细胞术检测血型糖蛋白a在细胞表面的表达。结果诃子酸和特里马素i在0.04～0.09？mmol／l浓度下均可显著抑制k562细胞的生长增殖。2种单宁化合物(0.002～0.01？mmol／l)可显著抑制丁酸钠诱导的k562细胞血红蛋白合成，2种单宁化合物(0.01～0.05？mmol／l)还可显著抑制氯化高铁血红素诱导的血红蛋白合成，特里马素i(0.01？mmol／l)还抑制丁酸钠诱导的gpa在细胞表面表达。结论诃子酸和特里马素i对红系分化有抑制作用。

The experiments of the biological activity for target molecula were accomplished. The experiment results of inhibiting activity against COX-2 indicated that the compound TM-II-5f had the highest inhibition rate, up to 95.59%, and yet the compound TM-II-5g exhibits weakly inhibiting activity.

对目标产物TM-II-5a~5g进行了生物活性研究，人环氧酶-2(COX-2)活性抑制实验结果表明：目标产物TM-II-5f对人环氧酶-2(COX-2)有很强的抑制活性，抑制率高达95.59%，目标产物TM-II-5g具有较弱的抑制率(0.61%)。

The results of bioassay experiments with 10 commonly used fungi showed that, all the title compounds had satisfactory fungicidal activity against Botrytis cinerea, the growth inhibition rate of compounds 5ae, 5ag, 5bd against Botrytis cinerea were up to 70% and for 5ad, 5cd, 5ce were more than 60%; compound 5bd exhibited fungicidal activity against Pellicularia sasakii with growth inhibition up to 60%, the growth inhibition rate of compound 5cg against Colletotrichum lagenarium was 69%.

抑菌活性生物测定结果表明，合成的大部分化合物对黄瓜灰霉病菌均有较好的生长抑制作用，其中，化合物5ae、5ag和5bd的抑制率达到70%；化合物5ad、5cd、5ce的抑制率大于60%；5bd对水稻纹枯病菌抑制率大于60%，化合物5cg对西瓜炭疽病菌的抑制率为69%。

Its activity was specific and was affected by pH, reaching the peak in weak acidic condition. It obviously inhibits amylases from D. melanogaster, Solenopsis invicta, Odontotermes formosanus, Periplaneta Americana Linnaeus, and Alphitobius sp. In addiction, the study points out Phaseolus vulgaris, Phaseolus coccineus L. and Glycine max, which have significant inhibition toward pancreatic amylase.

经测试发现此抑制剂在85℃时仍具备抑制果蝇淀粉酶之活性，为一热安定性蛋白质，其抑制作用受pH 值影响很大，在偏酸性环境下的效果最好，且其抑制作用具特性，可明显抑制果蝇、入侵红火蚁、白蚁、蟑螂及面包虫等昆虫的淀粉酶活性。

This conclusion is based on three groups of experiments with detached root tips of wheat seedlings: By following the time course changes of NO synthase , superoxide synthase and ABA accumulation under dehydration stress, we found that ABA accumulation was preceeded by the changes of NOS and superoxide synthase. ABA accumulation induced by dehydtrion stress and osmotic stress can be blocked by NO scanvegers and NOS inhibitors, while only dehydration stress-induced ABA accumulation can be blocked by ROS scanvegers. Exogenous applied NO or ROS induced ABA accumulation in root tips of wheat seedlings, and synergistic effects were found between NO and NO. The in planta expereiments also proved that ROS and NO are involved in water stress-induced ABA accumulation.Ⅱ.

证据主要来自以离体根尖为材料的实验：(1)通过检测干旱胁迫下小麦根尖NOS活性、O〓合成酶活性和ABA积累的时间变化进程，发现ABA积累滞后于ROS和NO的变化；(2)抑制剂实验表明，NO清除剂和NOS抑制剂可以抑制自然干旱胁迫及渗透胁迫诱导的小麦根尖ABA积累，ROS清除剂抑制自然干旱胁迫诱导的ABA积累而不抑制渗透胁迫诱导的小麦根尖ABA积累；(3)在非胁迫条件下施加外源的ROS或NO可以诱导小麦根尖积累ABA，ROS和NO之间具有协同作用。

The inhibition substances in Sorbus pohuashanensisHedl fruit not only restrained the seeds of wheat, cabbage from germinating but also restrained height and root growth. After the seeds of wheat, chinese cabbage had been soaked in the water extraction of pulp, seed and decoated seed for 8h, the seed germination rates were 92% and 84%, 89% and 65%, 94% and 78%, lower than the control, especially the water extract of decoated seed; and the root length and seedlings height were lower than the control, especially the water extract of pulp, and decreased in sequence of soaking time from short to long. So the simplest and effective method to eliminate pulp soluble inhibiting substances is to wash fruits by flowing tap water soon after collection.

在几种浸泡时间中，浸泡8小时的去皮种子浸泡液对白菜、小麦种子发芽率的抑制作用最为明显，其发芽率分别为65%、89%，但随着浸泡时间的延长而降低；浸泡8h的果肉浸泡液对白菜和小麦幼苗高生长和根伸长的抑制作用最为明显，种子和去皮种子浸泡液(8h)的抑制作用对小麦和白菜的抑制作用次之，随着浸泡时间的延长，果肉浸泡液的抑制作用逐渐减弱，因而采收下来的果实及时净种是清除果肉水溶性抑制物质简单有效的方法。

Results showed that the activity of soil poly-phenol oxidases and acid phosphatase, and soil respiration were suppressed by Starane at 0.5 and 5 mgkg^(-1) dry soil, respectively, during the first several days of experiment, but were slight promoted thereafter. In contrast, treatment with Starane at 50 mgkg^(-1) stimulated at the beginning of experiment but inhibited following that time the activity of soil poly-phenol oxidases and acid phosphatase and soil respiration. Activity of urease was stimulated at the beginning but inhibited in the following days by Starane at 0.5 and 50 mgkg^(-1) dry soil, respectively. However, the pattern of stimulation of urease activity at first several days of experiment followed by reduction to the basil level was observed. With respect to invertase, its activity was constantly depressed in the presence of Starane.

结果表明使它隆在0.5mgkg^(-1)和5mgkg^(-1)质量分数时对土壤多酚氧化酶、酸性磷酸酶和呼吸强度的影响为轻微抑制－激活－恢复稳定的趋势，50mgkg^(-1)质量分数时为轻微激活－抑制－恢复稳定的趋势；使它隆在0.5mgkg^(-1)和50mgkg^(-1)质量分数时对土壤脲酶活性的影响为激活-恢复稳定的趋势，5mgkg^(-1)时则处于抑制－激活的趋势；各质量分数的使它隆浓度对土壤蔗糖酶和土壤全酚均为抑制作用，且质量分数越大抑制越强烈。

According to the clear water experiment, aeration performance of the new equipment is good with high total oxygen transfer coefficient and oxygen utilization ratio.

曝气设备的动力效率在叶轮转速为120rpm～150rpm时取得最大值，此时氧利用率和充氧能力也具有较高值。

The environmental stability of that world - including its crushing pressures and icy darkness - means that some of its most famous inhabitants have survived for eons as evolutionary throwbacks, their bodies undergoing little change.

稳定的海底环境─包括能把人压扁的压力和冰冷的黑暗─意谓海底某些最知名的栖居生物已以演化返祖的样态活了万世，形体几无变化。