唑

The bioassays showed that the inhabitation rate of the mixture of two isomers, Z isomer and E isomer were reached 95%, 100% and 97% against Sphaerotheca fuliginea at 50 mg/L. The inhabitation rate of them was similar, so the mixture of the two isomers can be used without separation.

结果表明，当处理剂量为50 mg/L时，氯苯肟唑、Z-氯苯肟唑和E-氯苯肟唑的防效分别为95%、100%和97%，三者活性基本相当，故在实际中无须将两个异构体分离，混合体可直接应用。

The comparison test of this new methodwith spray inoculation method was conducted. The results showed the former method could increase the incidence ofdisease and uniformity than the latter one. Used cotyledon-brushing with conidial suspension and fungicide foliarspraying method, the EC 50 values of hexaconazole, myclobutanil, triadimefon, thiophanate-methyl and chlorotha lonil to Sphaerotheca fuliginea treated in different time after inoculation were determined; the results showed that 96 h was better time for disease severity evaluating.

比较了白粉病菌分生孢子悬浮液涂抹法和喷雾法接种黄瓜幼苗子叶的效果，结果表明，涂抹法发病率高，均匀度更好；测定了接菌后不同时间施药，白粉病菌对己唑醇、腈菌唑、三唑酮、甲基硫菌灵和百菌清等 5 种杀菌剂的敏感性，结果表明，接菌后 96h 施药较为敏感，测得的 EC 50 较小。

As for the ester exchange reaction on phosphorus, it was found that N-phosphoryl histidine the fastest one among all of the N-phosphoryl aminoacids. The results studied by MNDO method indicate that due to theparticipation of imidazole group, the formation of hexa-coordinatephosphorus intermediate made the iso-propoxyl which is opposite toimidazole group more active than the other ones and much easier to leave.When iso-propoxyl left, a new penta-coordinate phosphorus intermediate wasformed, and it is sterically favorable to be attacked by an alcohol from theopposite direction of imidazole.

对于磷上酯交换反应，实验中发现N-磷酰组氨酸反应速度明显高于其它N-磷酰氨基酸，理论研究表明，侧键咪唑基参与下六配位磷中间体形成后，位于咪唑基对面的异丙氧基反应活性大大提高，即从咪唑基的对面位置发生异丙氧基的离去和另一分子醇的进攻，在能量上和空间上都是有利的。N-磷酰丝氨酸的磷上酯交换反应有着类似的特点。

Methods of eating metronidazole along with 20% for part of burn is recommended to be used in treatment. Key words: Metronidazole; 20% of silver nitrate; Recurrent stomatologist RAU

笔者于临床上用甲硝唑（又名灭滴灵、甲硝哒唑、甲硝基羟乙唑）内服配合局部用20%硝酸银溶液点灼，治疗阿弗他性口炎128例进行跟踪观察，收到较理想的效果，而临床上未见有资料报道。

A convenient method to synthesize three kinds of novel 2-(2-hydroxyphenyl) benzimidazole in order to improve the solubilities of the fluorophores with substituent of carboxyl, ester and double-bond which are aimed for determining the sulphydryl group was reported.

合成了N-{3-(2-苯并咪唑基)-4-羟基苯基}马来酰亚胺酸， N-{3-(2-苯并咪唑基)-4-乙酸酯基苯基}和马来酰亚胺N-{3-(2-苯并咪唑基)-4-羟基苯基}马来酰亚胺，在基本荧光发射团上分别引入了羧酸基；酯基；双键活性基团。

High doses of fluconazole, itraconazole, and ketoconazole have been reported to be teratogenic in rodents.

有报道说高剂量的氟康唑、伊曲康唑和酮康唑在啮齿类动物可致畸形。

Author had started the research on design and synthesis of heterocycles several years ago, mainly focused on the design and synthesis of imidazole, thiazole, tetrazole derivatives and their glucosides, in which most of them may have some particular bioactivities.

本论文主要是围绕具有生理活性含氮杂环化合物的设计与合成而展开的，在论文工作中我们应用液相&一锅法&和固相组合化学方法进行了咪唑环、噻唑环、四氮唑环等具有生理活性的杂环化合物及其糖苷的合成。

Their tribological properties in paraffin and water were investigated with a four-ball test machine, the results shown that the thiadiazole derivatives and the imidazoline borates have better friction reduction and antiwear properties, and the thiadiazole derivatives also have excellent extreme pressure properties in water.

通过在四球摩擦磨损试验机上评价上述两类衍生物分散在液体石腊及水中的抗磨减摩性能，首次发现噻二唑及咪唑啉衍生物在水中也有较好的抗磨减摩性能，且噻二唑衍生物在水中具有良好的极压性能。

In this study, new benzo[l,2,3]thiadiazole derivatives were designed according to relationship of structure and efficacy. The 9 novel compounds were synsthesized with following reactions. The chlorine atom in 2-chloro-3,5-dinitro-benzoic acid as beginning raw material was substituted by 2-methylpropane-2-thiol, esterified then with bromoethane, reduced by iron powder and cyclized to obtain ethyl benzo[l,2,3]thiadiazole-7 after diazonation reation.

本论文根据苯并噻二唑诱导剂的构效关系设计了新的苯并噻二唑的结构，并合成了9个未见文献报道的化合物，合成步骤如下：采用2-氯-3，5-二硝基苯甲酸为起始原料，苯环上的氯原子被叔丁基硫醇置换，羧酸由溴乙烷酯化，硝基由铁粉还原，随后经重氮化关环生成苯并[1，2，3]噻二唑-7-羧酸乙酯。

Ivermectin shows similar effect on Ascaris with albendazole, better effect on Trichuris and poorer effect on hookworm and Enterobius than albendazole.

结论伊维菌素治疗鞭虫感染疗效优于阿苯达唑，治疗蛔虫感染疗效与阿苯达唑相同，治疗钩虫、蛲虫感染疗效不及阿苯达唑。

However, as the name（read－only memory）implies, CD disks cannot be written onorchanged in any way.

然而，正如其名字所指出的那样，CD盘不能写，也不能用任何方式改变其内容。

Galvanizes steel pallet is mainly export which suits standard packing of European Union, the North America. galvanizes steel pallet is suitable to heavy rack. Pallet surface can design plate type, corrugated and the gap form, satisfies the different requirements.

镀锌钢托盘多用于出口，替代木托盘，免薰蒸，符合欧盟、北美各国对出口货物包装材料的法令要求；喷涂钢托盘适用于重载上货架之用，托盘表面根据需要制作成平板状、波纹状及间隔形式，满足不同的使用要求。