化合物

Target compounds have been synthesized by condensation of the aromatic nucleus and amino heterocylcle with acyl isocyanates or acylisothiocyanates in absolutely anhydrous and aprotic solvent.

为了寻找高活性的农药品种，利用生物等排原理和亚结构连接法，对脲类化合物的母体结构进行了修饰，将芳氧羧酸类及吡唑环引入酰基脲母体结构中，利用酰基异氰酸酯与杂芳环胺类化合物在无水非质子溶剂中发生亲核加成反应，合成了四个系列21种新的酰基脲类目标化合物。

The anti-inflammatory activity of five of these compounds (B1, B4, B5, B6 and B7) was tested on mouse ear edema induced by croton oil, and the result showed that the inhibition ratios of compounds B4, B6 and B7 were between 65. 9%, 61. 7%and 52. 5%respectively (P.001%compared with control group), when the hypodermic injection dose was 50mg/kg, which are worthy for further research and development.

测定了其中5个化合物B1、B4、B5、B6和B7的抗炎活性（剂量为50mg／kg，皮下注射），发现化合物B4、B5和B7抗炎活性较好，对小鼠耳廓肿胀的抑制率分别为65.9％、61.7％和52.5％，和对照组相比P.001，这些化合物有进一步研究开发的价值。

Hydroxynitrilelyase, a vital tool in the bio-synthesis of optically active cyanohydrin, which can catalyze carbonyls and HCN selective forming optically active cyanohydrin.

醇腈酶(α-hydroxynitrilelyase， HNL)是手性醇腈化合物生物合成十分有用的工具，能够催化羰基化合物和HCN立体选择性的加工形成手性醇腈化合物。

The present invention relates to the depolymering cyclization reaction of aromatic dithio ether polymer to prepare aromatic cyclic dithio ether compound under the presence of mercapto group containing compound and alkali matter.

本发明涉及利用芳香双硫醚聚合物的解聚成环反应来制备芳香双硫醚环状化合物的方法。该方法采用芳香双硫醚聚合物在含巯基的化合物和碱性物质存在的条件下发生解聚成环反应生成双硫醚环状化合物。

The reaction of polyfluoroalkyl iodides with 4-pentenoic acids initiated by sodium dithionite was realized to give polyfluoroalkyl substituted lactones.

我们研究了多氟烷基碘代烷与4-戊烯酸类化合物等在连二亚硫酸钠引发下的反应，得到了氟烷基取代的内酯化合物，我们将该反应称为氟烷基化内酯化反应；并建立了一个利用该反应合成含氟内酯的新方法，首次利用氟烷基化内酯化反应进行高立体选择性双环含氟内酯及手性含氟内酯等的合成，已合成含氟内酯新化合物50余种。

In chapter 2, the contents of loureirins in the roots, stems and leaves of Dracaena cochinchinenis were analyzed by HPLC. On the other hand, using the preparation chromatography technology, five compounds were isolated from the leaves of Dracaena cochinchinenis, their structures were identified by means of spectral and chemical methods. They are steroidal saponins.

第二章主要是利用HPLC技术对剑叶龙血树根、茎、叶中龙血素成分的分析与探讨，并利用制备色谱等技术对剑叶龙血树叶子组成成分进行了分析、研究，得到化合物5个，经波谱鉴定，这5个化合物均是幽体皂贰类化合物。

The compound is an ionic compound consisting of a cation NH(subscript 4 superscript +) and an anion C6H2N3O(subscript 9 superscript -), and it is the mono-substituted salt of TNPG. Since the existence of complicated hydrogen bond networks and electrostatic attraction between NH(subscript 4 superscript +) cation and C6H2N3O(subscript 9 superscript -) canion, the compound possesses better stability and low sensitivity.

该化合物是由一个铵根离子与一个一价的三硝基均苯三酚负离子相结合而形成的离子型化合物，分子中存在的大量氢键及铵根离子与三硝基均苯三酚负离子之间的静电引力使得该化合物具有较高的热稳定性和较低的感度。

Compounds 1 and 2 were new compounds, compounds 3 and 9 were isolated from this genus for the first time.

其中化合物1和2为新化合物，化合物3和9为首次从该属植物中分离得到。

The essential oil was prepared from the peel by solution extraction, and separated into fractions of hydrocarbon and oxygenated compounds through a silicagel column. As the oxygenated fraction had the characteristic aroma of the peel oil, odor quality of the fraction was estimated on the basis of a odor unit value. Twenty five compounds such as geranial, neral, linalool and aliphatic aldehydes were selected as the components contributed to the aroma of the peel oil.

用溶剂萃取法提取白柠檬果皮的精油，并用硅胶柱将精油分成碳氢化合物和含氧化合物两大部分，由于含氧化合物部分具有果皮油的特征香气，利用各成分的香气值对该部分进行了评价，明确了香叶醛、橙花醛、沉香醇以及一些脂肪族醛等25种成分对白柠檬果皮油香气起着重要作用。

OBJECTIVE: Three sesquiterpene lactones 1-O-acetylbritannilactone, isoalantolactone and britannilactone were isolated from the roots of Inula helenium and the flowers of Inula japonica. The antitumor activities of the three sesquiterpenoids in the cell lines of HeLa, HEC-1, SHIN3, HOC-21 and HAC-2 were measured, and the relationship between structure and activity and the possible mechanisms were explored.

目的： 观察菊科植物中分离出的3种倍半萜化合物异土木香内酯、1-氧-乙酰大花旋覆花内酯和大花旋覆花内酯对体外培养的人子宫颈癌HeLa细胞、人子宫内膜癌HEC-1细胞、人卵巢透明细胞癌SHIN3及HOC-21细胞和人卵巢囊腺癌HAC-2细胞增殖的影响，研究这3种倍半萜化合物的体外抑制肿瘤细胞增殖作用及其结构与活性之间的构效关系，进而探讨3种倍半萜化合物的体外抑制肿瘤细胞增殖的可能机制。

The split between the two groups can hardly be papered over.

这两个团体间的分歧难以掩饰。

This approach not only encourages a greater number of responses, but minimizes the likelihood of stale groupthink.

这种做法不仅鼓励了更多的反应，而且减少跟风的可能性。