乙酰氯

The most commonly used drugs Bleomycin, mitomycin C, Adriamycin, 5 - 5-fluorouracil (5 - Fu), methotrexate, cyclohexyl - nitrosourea, imipramine hydrazone, Vindesine, etoposide (VP-16), chlorine and ammonia-platinum, a single chemotherapy drug remission rate in the 15% to 20% remission for 1 to 4 months.

最常用的药物有博来霉素、丝裂霉素C、阿霉素、5-氟尿嘧啶（5-Fu）、甲氨喋呤、环己亚硝脲、丙咪腙、长春花碱酰胺、鬼臼乙叉甙（VP-16），以及顺氯氨铂，单一药物化疗的缓解率在15％～20％，缓解期为1～4个月。

ResultThe Buxus Microphylla leaf ethyl acetate extraction (high-dose and low dose) have obvious effect on reducing the serum total cholesterol and triglyceride, moreover, the high-dose ethyl acetate extract reducing blood lipid was better than the other extracts.

结果 小叶黄杨叶乙酸乙酯提取物的高、低两个剂量组均有显著的降低血清总胆固醇和三酰甘油的作用，小叶黄杨叶的水提取物和石油醚提取物均有显著的降低血清中总胆固醇的作用，小叶黄杨叶氯仿提取物及正丁醇提取物均无降血脂的作用。

The new surfactant was synthesized from the main starting materials such as lauric acid, p-cresol, chlorosulphonic acid and ethylene diamine, by 5 classic reactions which are acyl chlorination, esterification, Fries rearrangement, sulfonation and condensation, with total yield of 58%.

作者以十二酸、对甲酚、氯磺酸、乙二胺等为主要原料，共采取了酰氯化、酯化、Fries重排、磺化和缩合等5步经典的单元反应，合成了该表面活性剂，总收率为58％，并探讨了各步反应的条件对收率的影响。

Four new salicylaldehyde derivatives with a glucose or mannose moiety were synthesized with 2-tert-butylphenol or 4-tert-butylphenol as the starting material, followed by the formylation, chloromethylation, nucleophilic substitution reaction with the desired carbohydrate. The salicylaldehyde derivatives condensed with ethylenediamine to give the Schiff bases, which coordinated with Mn to afford four novel sugar-based Salen Mn complexes.

首先，分别以2-叔丁基苯酚和4-叔丁基苯酚为起始原料，经过甲酰化反应、氯甲基化反应、和糖类衍生物的亲核取代反应制得了四种新型并入葡萄糖基或甘露糖基的水杨醛衍生物，将它们与乙二胺缩合生成希夫碱配体，得到的配体与过渡金属Mn~(3+)配位制备出四种新型含糖基的Salen Mn配合物。

A key intermediate of abacavir, named N-(2-amino-4,6-dichloro-5-pyrimidinyl) formamide was synthesized from diethyl malonate and guanidine hydrochloride. This method suits to industry for large scale. The materials are easy to get and very cheap.

2-氨基-4，6-二氯-5-甲酰氨基嘧啶是合成阿巴卡韦的关键中间体，本文拟以丙二酸二乙酯和盐酸胍为起始原料合成这一关键中间体，具有原料来源广，适合大规模生产等优点。

Following resolution, the following steps are performed: reduce the isomer to an alcohol, react the alcohol with triphenylmethyl chloride, ozonalyze the resulting reaction product, reduce the ozonalyzed product to yield a diol and react the diol with a methane sulfonyl compound to form-3-2-{(methylsulfonyloxy}ethoxy-4--1-butanol methane sulfonate.

拆分后，进行下一步：将异构体还原为醇，使醇与三苯基甲基氯反应，臭氧化所得反应产物，还原臭氧化产物以得到一种二醇并使所述二醇与甲烷磺酰基化合物反应以形成-3-2-{(甲基磺酰基氧}乙氧基-4--1-丁醇甲烷磺酸酯。

The solubility of the novel polyamides are greatly improved compared with the conventional aramids, especially the polyamide with dendritic blocks of the second genernation as side chains are soluble in most of the common organic solvents such as ether, ethyl acetate, chloroform, acetone, tetrahydrafuran etc.

树状片段的引入大大地改善了聚酰胺的溶解性，特别是以第二代树状片段为侧基的聚酰胺的溶解性得到了很大的改进，可以溶于大部分常见的有机溶剂，如乙醚、乙酸乙酯、氯仿、丙酮、四氢呋喃等。

To synthesize aryl pyrimidines by taking benzene, methyl benzene ,acetic ether,1,2-dichloroethane as solvent,the yield and purity of the product are high by taking methyl benzene as solvent.

分别选用苯、甲苯、乙酸乙酯、二氯乙烷作为溶剂合成桂皮酰哌啶，结果表明甲苯作为溶剂时产品纯度高，收率高，可用于大规模生产。

Three methods for the preparation of 1,2,4-trizolone~5 are provided. 22 compounds are prepared. 3, 4-disubstituted 1,2,4-trizolone-5 is prepared by reacting amide with ethyl hydrazine-fornate at 110癈 for 3h in the presence of phosphorus oxychloride, following neutralization and cyclization reaction, giving to 74.5 % yields,which is 30% more than the literature value.

以三氯氧磷为缩合剂，使酰胺和肼基甲酸乙酯在110℃反应3h，经碱中和、环化反应，合成3，4-二取代-1，2，4-三唑酮-5，两步反应总产率达74.5％，与文献报道值相比，高出了30％以上，在三唑酮类衍生物的合成方法中具有很大的突破性。

According to the clear water experiment, aeration performance of the new equipment is good with high total oxygen transfer coefficient and oxygen utilization ratio.

曝气设备的动力效率在叶轮转速为120rpm～150rpm时取得最大值，此时氧利用率和充氧能力也具有较高值。

The environmental stability of that world - including its crushing pressures and icy darkness - means that some of its most famous inhabitants have survived for eons as evolutionary throwbacks, their bodies undergoing little change.

稳定的海底环境─包括能把人压扁的压力和冰冷的黑暗─意谓海底某些最知名的栖居生物已以演化返祖的样态活了万世，形体几无变化。