-甲基哌啶

Results There were 22 lacunar infarction cases, 1 case large area infarction, and 8 cases with small bleeding in the thalamus, 1 case with large bleeding in the basal ganglia of 9 cases intracerebral hemorrhage. Hemichorea appeared in 27 cases within 24 hours, 5 cases within 1 week. All received aloperidin, the symptom disappeared in27 cases（84.4%）.

结果 32例偏侧舞蹈症病例中脑梗死23例(腔隙性脑梗死22例，大面积脑梗死1例)，脑出血9例(丘脑少量出血8例，基底节区大量出血1例)；脑卒中后24h与1周内出现偏侧舞蹈症症状分别为27例和5例；应用氟哌啶醇治疗后症状消失27例。

The patients can appear hemichorea when he had cerebral infarction with Basal ganalia injury symptoms of them can be controlled by Haloperidol and Nitrazepam.

节论 损伤基底神经节的脑梗死可以出现偏侧舞蹈病，氟哌啶醇和硝基安定可以控制其症状。

Treatment with dopamine and low dose bromocriptine resulted in cell death accompanied with the DNA laddering and activation of caspase-3 only in GH3D2L and GH3D2S cells, which were blunted by haloperidol, showing that dopamine-induced cell death in these cells is mediated by dopamine D2 receptors.

经多巴胺和低浓度溴隐亭处理后仅在GH3D2L和GH3D2S两种细胞中出现细胞死亡伴DNA阶梯状断裂和半胱天冬酶3（Caspase-3）的激活，而这些效应也被氟哌啶醇所抑制，说明多巴胺所致的细胞凋亡与多巴胺D2受体激活有关。

Neu- roleptics such as Haloperidol and Tiapide might increase theta waves of the anterior and medius areas of the head of brain electrical back- ground activity of children with TS, and affect their memory func- tion, but not affect their intelligence, personality and behavior.

氟哌啶醇和泰必利等精神抑制药物可能使TS患儿头前中部区域的脑电背景活动θ波增多；并对TS患儿的记忆功能可能产生一定的影响，但对TS患儿的智力、个性和行为无明显影响。

It suggested neuroleptics such as Haloperidol and Tiapide might increase theta waves of the anterior and medius areas of the head of children with TS.

用药组头前中部区域（前额区、额区、中央区和顶区）θ频段分布百分比显著多于对照组，提示氟哌啶醇和泰必利等精神抑制药物可能使TS患儿头前中部区域的脑电背景活动θ波增多。

Moreover, the preliminary test of the biological activity of the 8 target derivatives showed that 7-(2-adenine)ethoxyl-2-ethyl-4"- methoxy isoflavone and 7-(2-hydroxyl-3-piperidino)propoxy-2-ethyl-4"- methoxyl isoflavone have fine biological activities on suppression of the growth of MCF-7 cell in breast cancer and the hela cell in cervical cancer of human being.

另外还对8个目标衍生物进行了初步的药理活性试验，发现7-(2-腺嘌呤)乙氧基-2-乙基-4′-甲氧基异黄酮和7-(2-羟基-3-哌啶)丙氧基-2-乙基-4′-甲氧基异黄酮均有较好的抑制人乳腺癌MCF-7细胞和人宫颈癌hela细胞生长的药理活性。

Haloperidol but not sulpiride enhanced the paired-pulse inhibition elicited by antidromic -orthodromic paired-pulse stimulation, and reduced the paired-pulse fa- cilitation evoked by orthodromic paired-pulse stimulation.

氟哌啶醇加强逆-顺向双脉冲刺激诱发的双脉冲抑制，减弱顺向双脉冲刺激诱发的双脉冲易化。

The final product Rimonbant was then obtained in 64% yield via chlorination of the acid with oxalyl chloride followed by treatment of the resultant acyl chloride with 1-aminoperidine.

酰氯与1-氨哌啶在三乙胺存在下缩合生成目标产物利莫那班，产率64%。

Fourteen unreported N-substituted piperidin-4-one oxime ethers derivatives were synthesized withsubstituted benzylamines or phenethylamine as raw materials via a series of Michael addition, Dieckmann condensation, hydrolysis decarboxylation reactions, oximation a...

以取代苄胺或苯乙胺为起始原料，依次经Michael加成，Dieckmann缩合，水解脱羧，肟化和醚化等多步反应合成了14个未见文献报道的N-取代哌啶酮肟醚衍生物。

We screened a set of Lewis base organocatalysts derived from chiral pipecolinic acid and tert-butanesulfinamide for the reduction of-N-Cbz-1- phenylpropenamine, including newly designed ones and some of those previously developed in our lab. However, only moderate stereoselectivities, albeit high yields were obtained.

在本课题组前期研究的基础上，我们筛选并设计了一系列以手性哌啶酸和叔丁基亚磺酰胺为母体的有机小分子路易斯碱催化剂，它们能催化三氯氢硅对-N-苄氧羰基-1-苯基丙烯胺的不对称还原，获得很高的收率和中等的对映选择性，并且具有很好的底物普适性。

The basic concept of FOP can be summarized as to further optimize effective prescription according to the standard of curative effects and with the aid of modern science and technology and theories of traditional Chinese medicine.

其基本内涵可概括为：以确有疗效的中药复方为研究对象，以现代科学技术和传统中医药理论为技术支持，以该复方所治病证的药效响应为评价标准，以优化重组疗效更优的新复方为研究目的。

Ever since our world has been a world, native forests have been indiscriminately exploited by man.

自从我们的世界一直是世界原生森林被任意剥削人。