查询词典 more active

These studies indicate the rationality of our molecular design based on the crystal structure of KARI complex. To obtain more KARI inhibitors with high activities, the molecular docking and 3D-QSAR methods were applied to our further studying of these amidine compounds. Two methods AutoDock3. 0.3 and DOCK4. 0 were used in molecular docking, and the calculate results accord with that of herbicidal tests in general. The CoMFA model from 3D-QSAR analysis provided useful guidance for designing highly active compounds prior to their synthesis.

这些分子作为潜在的KARI抑制剂为基于KARI的农药分子设计提供了有利指导；对部分小分子进行了合成，在除草活性初筛的近三十个化合物中，个别化合物表现出较好的除草活性，其中一个化合物wb1596对油菜和稗草具有较高的生长抑制率，并通过E.coli KARI酶活性抑制试验验证了其KARI酶的作用靶标，此化合物可以作为KARI一个有苗头的抑制剂为后续工作奠定了基础；对发现的有苗头的KARI抑制剂进行了结构修饰和优化，合成了一系列脒类化合物并确证了它们的结构，改造后的化合物与原抑制剂相比大多除草活性相当或更佳，从而表明我们基于靶标结构的分子设计的合理可靠性；对所合成一系列脒类化合物进行了分子对接和三维定量构效关系研究。

In aqueous solution no binding observed in crystal structure. In cyclohexane, one amylamine molecule is observed in the active site of trypsin and more sulfates are also found on enzyme surface, which are further proofs that electrostatic interaction are stronger in organic solvent.

在水溶液中，晶体结构难以观察到戊胺与牛胰酶的结合，在环己烷中，一个戊胺分子结合在胰酶的活性中心，同样酶表面观察到了更多的硫酸根，这些都进一步验证了有机溶剂中静电相互作用加强。

Peripheral neutrophils are activated in anaphylactoid purpura, which seems to be more obvious in active phase than in remission phase.

过敏性紫癜患者外周血中性粒细胞处于激活状态，活动期较缓解期更明显。

Antituberculosis treatment is complicated by frequent drug-interactions with highly active antiretroviral therapy and adverse drug reactions are more common among HIV-infected patients.

抗结核药物与高效抗逆转录病毒药物的副作用及时常发生的相互作用使得HIV-TB合并感染的治疗更趋复杂化。

Light curing speed by up to 100 ~ the giant 300 m/min; and 3 with the UV glazing process on the business card printing and membership card production, color much later than other artifactitious attractiveto stays fresh and cured coatings and wear-resistant, more resistant to the drug resistance and chemical resistance, good stability, be able to wash water and ethanol; 4 to UV on volatile high active ingredients, so the relatalion province.

灯照射下固化速度可达100~300m/min； 3经UV上光工艺处理后的制卡和会员卡制作品，色彩明显较其他加工方法鲜艳亮丽，而且固化后的涂层耐磨，更具有耐药品性和耐化学性，稳定性好，能够用水和乙醇擦洗； 4UV上光油有效成分高，挥发少，所以用量省。

Even more, since it has the active substance of natural berbal medicine, whiceh can permeate into the conified layer of skin, it can clean the detrimental substances, and kill the bacteric and virus.

它含有昆达---2号生物淬取液和名贵香料、维生素、天然保湿分子、蜂王浆等多种营养成份，使其不仅具有气味清新、泡沫丰富、润肤养颜等特点，更因其含有天然药用植物的活性物质，可深入人体皮肤角质层，清除有害物质，杀灭病菌，对由真菌引起的脚气、湿疹、体等皮肤病具有奇特的治疗效果。

Even more, since it has the active substance of natural berbal medicine, whiceh can permeate into the conified layer of skin, it can clean the detrimental substances, and kill the bacteric and virus.

它含有昆达---2号生物淬取液和名贵香料、维生素、天然保湿分子、蜂王浆等多种营养成份，使其不仅具有气味清新、泡沫丰富、润肤养颜等特点，更因其含有天然药用植物的活性物质，可深入人体皮肤角质层，清除有害物质，杀灭病菌，对宫颈糜烂有显著的辅助疗效、对由真菌引起的脚气、湿疹、体等皮肤病具有奇特的治疗效果。

So-called banausic work, which included manufacturing, business, and trade (which were not tied to the land and the family farm), and what we would call "capitalism"(investing money to make more money) were considered to be incompatible with active participation in the affairs of the polis and even as unnatural and morally corrupting.

所谓事物的工作，其中包孕制造业，商业和贸易（其中无关的土地和家庭大农场），和我们所称的&资本主义&被以为是不符合积极参与国际事件的城邦，甚至不自然和道义上的腐败。

So-called banausic work, which included manufacturing, business, and trade (which were not tied to the land and the family farm), and what we would call "capitalism"(investing money to make more money) were considered to be incompatible with active participation in the affairs of the polis and even as unnatural and morally corrupting.

所谓物质的工作，其中包括制造业，商业和贸易（其中无关的土地和家庭农场），和我们所称的&资本主义&被认为是不符合积极参与国际事务的城邦，甚至不自然和道义上的腐败。

About 250 hourly employees have been recalled to the smelter in recent days, boosting its total active work force to more than 400, including about 100 workers at the billet casthouse.

最近几天，工厂已经召回了250名小时工人，工厂劳动力增至400多名，其中包括铝锭铸造车间的100名工人。

We have no common name for a mime of Sophron or Xenarchus and a Socratic Conversation; and we should still be without one even if the imitation in the two instances were in trimeters or elegiacs or some other kind of verse--though it is the way with people to tack on 'poet' to the name of a metre, and talk of elegiac-poets and epic-poets, thinking that they call them poets not by reason of the imitative nature of their work, but indiscriminately by reason of the metre they write in.

索夫农 、森那库斯和苏格拉底式的对话采用的模仿没有一个公共的名称；三音步诗、挽歌体或其他类型的诗的模仿也没有——人们把&诗人&这一名词和格律名称结合到一起，称之为挽歌体诗人或者史诗诗人，他们被称为诗人，似乎只是因为遵守格律写作，而非他们作品的模仿本质。

The relationship between communicative competence and grammar teaching should be that of the ends and the means.

交际能力和语法的关系应该是目标与途径的关系。