查询词典 inhibitors

The firing patterns induced by veratridine and aconitine, inhibitors of inactivation gate of sodium channel operating on different binding sites, were compared.

藜芦碱和乌头碱是钠通道失活门的抑制剂，但二者作用于不同的位点，前者结合于D2-S6，后者结合于D3-S6。我们比较了这两种试剂引发的放电模式。

PS developering is mainly composed of reagents, inhibitors and wetting agent.

PS版显影液主给由显影剂、抑制剂以及湿润剂构成。

AIM: To investigate the prerequisite of the integrated method for characterizing inhibitors with the inhibition of xanthine on Candida species uricase as the model.

目的：以Candida species尿酸酶为模型，考察用积分法筛选抑制剂的条件。

Based on analyses of the present applications of corrosion inhibitors for recirculated cooling water, a new-type of complex corrosion inhibitor containg molybdate, zincate, organic acid and gluconate was proposed.

为解决某水样的腐蚀问题，提出了一种由钼酸盐、锌盐、有机酸、葡萄糖酸盐等组分的复合缓蚀剂配方，设计了正交实验，并采用旋转挂片测定了其腐蚀速度。

This process is the result of the imbalance between matrix metalloproteinases zymogen activations and interaction of the active forms with specific tissue inhibitors of metalloproteinases.

本实验以大鼠为模型旨在研究急性胰腺炎中基质金属蛋白酶-2(MMP-2)与基质金属蛋白酶特异组织抑制物-2(TIMP-2)在胰腺组织中的表达，探讨其与急性胰腺炎时器官损伤程度的相关性。

The aconitic acid-acrylic acid copolymer, itaconic acid homopolymer and polyepoxysuccinic acid which were non-phosphorus scale and dispersing inhibitors were synthesized with the fermentation products citric acid, itaconic acid and maleic anhydride.

以生物发酵产品柠檬酸和衣康酸为主要原料，分别合成了无磷阻垢分散剂丙烯三羧酸－丙烯酸共聚物和衣康酸均聚物，利用马来酸酐合成了聚环氧琥珀酸。

The structure reveals the catalytic intermediate of DAPDC, in which L-lysine is covalently bonded to PLP to form an external aldimine. This conformation provided the best insight to date on the substrate binding and catalytic mechanism of DAPDC. It also supplied valuable clues for designing specific DAPDC inhibitors.

通过分析我们发现这是DAPDC酶家族的第一个反应中间态结构，即反应产物L-赖氨酸与辅酶PLP共价结合形成了外源醛亚胺的构象，这为了解DADPC的底物结合情况及催化机理提供了迄今为止最详细深入的结构信息，也为针对DAPDC设计特异性抑制剂提供了宝贵的线索。

These studies indicate the rationality of our molecular design based on the crystal structure of KARI complex. To obtain more KARI inhibitors with high activities, the molecular docking and 3D-QSAR methods were applied to our further studying of these amidine compounds. Two methods AutoDock3. 0.3 and DOCK4. 0 were used in molecular docking, and the calculate results accord with that of herbicidal tests in general. The CoMFA model from 3D-QSAR analysis provided useful guidance for designing highly active compounds prior to their synthesis.

这些分子作为潜在的KARI抑制剂为基于KARI的农药分子设计提供了有利指导；对部分小分子进行了合成，在除草活性初筛的近三十个化合物中，个别化合物表现出较好的除草活性，其中一个化合物wb1596对油菜和稗草具有较高的生长抑制率，并通过E.coli KARI酶活性抑制试验验证了其KARI酶的作用靶标，此化合物可以作为KARI一个有苗头的抑制剂为后续工作奠定了基础；对发现的有苗头的KARI抑制剂进行了结构修饰和优化，合成了一系列脒类化合物并确证了它们的结构，改造后的化合物与原抑制剂相比大多除草活性相当或更佳，从而表明我们基于靶标结构的分子设计的合理可靠性；对所合成一系列脒类化合物进行了分子对接和三维定量构效关系研究。

Which of the following statements could be most likely to come after the last sentence of the passage?+ b' C- _ e1 K% h \ ^0 f The failures of the past, however, must not impede further research into the amnestic action of protein-synthesis inhibitors.

在这个类比的例子之前，通篇都是在讲为什么人们觉得不是蛋白质合成来导致失忆，而没有明确提到是如何发现正确的理论。

The antiscale rates of LA and some common scale inhibitors were determined through the static scale inhibition method.

利用静态阻垢法测定和比较LA与一些常用阻垢剂的阻垢率。

According to the clear water experiment, aeration performance of the new equipment is good with high total oxygen transfer coefficient and oxygen utilization ratio.

曝气设备的动力效率在叶轮转速为120rpm～150rpm时取得最大值，此时氧利用率和充氧能力也具有较高值。

The environmental stability of that world - including its crushing pressures and icy darkness - means that some of its most famous inhabitants have survived for eons as evolutionary throwbacks, their bodies undergoing little change.

稳定的海底环境─包括能把人压扁的压力和冰冷的黑暗─意谓海底某些最知名的栖居生物已以演化返祖的样态活了万世，形体几无变化。