查询词典 inhibitor

U73122 and pyrrolidine dithiocarbamate (an inhibitor of NF-κB) were used to study the effect of PLCγ1 and NF-κB on cell-matrix adhesion.

吡咯二硫氨基甲酸酯用于研究NF-κB在结直肠癌细胞与基质黏附中的作用。

Methods Mouse macrophages were stimulated with Mpe LAMPs to analyze the activitation of NF-κB, and the effect of pyrrolidine dithiocarbamate, an inhibitor of NF-κB, on NF-κB activation was also studied by indirect immunofluorescence and western blot.

用从穿透支原体中提取的脂质相关膜蛋白刺激小鼠巨噬细胞，经Western blot和间接免疫荧光等方法检测NF-κB是否被激活，以及NF-κB抑制剂PDTC对NF-κB活性的影响。

In the poly-merization system,oxygen acted not only as the inhibitor of polymerization,but also as the quencher of the triplet of the initiator.

氧在Eo(IPh2)2光敏引发聚合中，既起自由基聚合阻聚剂的作用，又起引发剂三重态猝灭剂作用

Became higher when cell was treated by Staurosporine while they are lower when treated by Quinacrine or Verapamil.To identify when the cytoxic signal transducts into the plasma and the time efffects of various inhibitor after cytokines combinds with their receptors.

Staurosporine促进细胞凋亡的过程浙江大学硕士学位论文伴随着Caspases和 Caspase3活性的升g，u Qui删rine和 Veraparnil 在抑制细胞凋亡的过程中Caspases的活性变化不大，而Caspase3的活性则相应降低。

To investigated the relationship of the signal transduction pathway and other signal molucules, three signal transduction inhibitors were tested for their effects on L929 cell and the change of caspase activation. The inhitors include Staurosporine Quinacrine (PLA2 inhibitor) andVerapamil (Ca2+ channel blocker).

为了探讨γTNFβ和TNFβ诱导细胞凋亡的信号转导通路与其它信号分子的关系，我们检测了蛋白激酶C抑制剂Staurosporine、磷脂酶A2抑制剂Quinacrine和钙离子通道阻断剂Verapamil对γTNFβ及TNFβ杀伤L929细胞的影响及其伴随的Caspase8和Caspase3活性的变化。

The characteristics of quinazoline epidermal growth factor receptor inhibitors were briefly described in this paper, and the mechanism of receptor-tyrosine kinase inhibitor was also introduced. The synthesis of this kind of new compound was studied, and the synthetic route was redesigned and the method was modified.

本论文简述了受体酪氨酸激酶小分子抑制剂的发展概况，详细介绍了新型喹唑啉类表皮生长因子受体抑制剂，着重研究了该类化合物的合成，设计并打通了合成路线，同时又合成了25个新化合物。

Objective: through various chemical synthesis target compounds 4 -- 6 - the - 7 -(2 - hydroxyl replace c oxygen radicals) quinazoline compounds were synthesized and the structure of the modified, so as to get high epidermal growth factor receptor tyrosine kinase inhibitor.

目的：通过各种化学合成方法完成目标化合物4--6-甲氧基-7-(2-羟基取代丙氧基)喹唑啉的合成并对目标化合物进行结构修饰，以期获得高活性的表皮生长因子受体酪氨酸激酶抑制剂。

Special attention was directed toward finding inhibitors selective against KDR tyrosine kinase in order to ensure that the in vivo profile of a specific Src inhibitor could be determined. The 4-aminobenzodioxole quinazoline series gave compounds with excellent potency and selectivity.

一直以来，人们为了确保能够在体内测定Src酶专属性抑制剂的特性，把研究焦点放在对KDR酪氨酸激酶选择性的抑制剂的寻找上。4-氨基苯并间二氧五环喹唑啉系列化合物具有极好的效力和选择性。

The predicted complex structure of quinazoline type inhibitor with EGF-R, as well as the pharmacophore mapping from CoMFA, can interpret the structure-activities of the inhibitors well and afford us important information for structure-based drug design.

基于定量构效关系研究和复合物结构模型，我们对抑制剂的改造提出了一些新的思路。

Quinidine, an established inhibitor of CYP2D6, was used as the positive control.

奎尼丁，一个已经被证实对 CYP2D6抑制的化合物，被用来作为正面对照。

The X-ray diffract was used to analyze the crystal structure of the composite. Results show that after the talc was treated with blend coupling agent, the crystal structure of talc changed, and effect Intercalation phenomenon.

通过X射线衍射分析可知，用混合偶联剂对滑石粉进行预处理后，滑石粉晶体结构发生改变，产生了插层现象，使PP／滑石粉复合材料为纳米复合材料。

An authentic Maui wedding might require the services of a 'kahu', which is a Hawaiian minister.

毛伊可能需要一个真实婚礼服务'kahu'，这是夏威夷部长。