查询词典 benzamide

In search of safer and more effective fungicidal compounds,eight N-(4,6-disubstitued pyrimidin-2-yl)- benzamide s were designed and synthesized.

为了寻找高效、安全的杀菌活性化合物，设计并合成了8个N-(4，6-二取代嘧啶-2-基)苯甲酰胺类化合物，其化学结构经1HNMR、IR、LC/MS和元素分析确证。

The paper proposed a possible binding mode of MS-275, a benzamide histone deacetylase inhibitor, to HDAC by intensive docking study.

通过计算机模拟的对接过程研究，发现了MS-275--一种苯甲酰胺类的组蛋白去乙酰酶抑制剂与酶的可能的全新结合方式。

The results showed that the application of photocatalytic oxidation to the treatment of wastewater was feasible and efficient, but it was affected by the operation conditions.There existed optimum value of the dosage of catalyst, initial benzamide concentration and pH value for the photocatalytic oxidation performance.H2PO-4,Cl-, Cu2+ and Al3+ showed obvious inhibition to the photocatalytic oxidation.

结果表明，循环式浆态光催化反应器中光催化剂的用量、污染物的初始浓度和初始pH值对模拟污染物光催化降解性能的影响存在适宜值；体系中H2PO-4、Cl-、Cu2+、Al3+对其光催化降解过程有明显的抑制作用。

Four adduct compounds are found for the former, and three are found for the latter. This indicates the DNA adduct formation capabilities both of 2-chloro benzamide and the photoproduct sample. Meanwhile the result of Ames experiments of them is positive. Thus we should pay more attention to important meaning of these results since the compound, which can produce adducts with DNA, may possibly be tumorigen or even carcinogen and mutagen.

结果表明，前者与DNA反应形成四个可辨认的加合物斑点，后者与DNA反应形成三个可辨认的加合物斑点，能与DNA加合的物质为潜在的&三致&物质，同时，二者的Ames试验结果显阳性这应当引起人们对灭幼脲环境安全性的重视。

The mechanism of carbon-nitrogen coupling reaction of 2-Iodo-selenophene with benzamide catalyzed by CuI has been investigated with density functional theory at GGA/PW91/DND level. The geometric configurations of reactants, intermediates, transition states, and products were optimized and verified by means of vibration frequency calculations.

采用密度泛函理论方法，在GGA/PW91/DND基组与水平上研究了2-碘代硒苯与苯甲酰胺在CuI催化下的微观反应机理，优化了反应过程中的反应物、中间体、过渡态和产物。

The photocatalytic oxidation performance and kinetics of the simulated organic wastewater in a circulating slurry photocatalytic reactor was investigated.The effects of operation conditions, such as dosage of photocatalyst, illumination time, initial benzamide concentration, pH value, anions and cations in wastewater, on the photocatalytic oxidation performance were discussed.

采用循环式浆态光催化反应器对苯甲酰胺模拟废水光催化氧化特性和动力学进行了研究，系统地考察了操作条件对模拟污染物光催化降解的影响，并与搅拌式和鼓泡床式浆态光催化反应器中苯甲酰胺的降解效果进行对比。

The results showed that precursor feeding (phenylanine, sodium acetate and benzamide) and mixed sugar as production medium resulted in significant increase of taxol production not only in the one-liquid-phase cultures of Taxus chinensis var. mairei but also in the two-liquid-phase cultures. And the integrated function of precursor feeding and mixed sugar in the two-liquid-phase cultures gave more significant increase of taxol production significant increase of taxol production, which was four times more than that of the control (the one-liquid-phase culture without precursors and mixed sugar).

结果表明前体饲喂（苯丙氨酸，醋酸钠和苯甲酰胺）和蔗糖与麦芽糖配伍作为生产培养基糖源不仅对红豆杉细胞悬浮培养，而且对其两液相培养的紫杉醇产量提高均有明显的促进作用，与对照组相比，在南方红豆杉细胞两液相培养中，采用前体饲喂和蔗糖与麦芽糖配伍作为生产培养基糖源，紫杉醇产量提高4倍多。

A transformant line obtained by transfection of NTH3T3 cells with c-Ha-T24-ras gene was treated with 5mmol/L benzamide,an inhibitor of PARP enzyme for 4 weeks.Some changes in cellular properties of the transformant line were observed.

用 5mmol/L PARP抑制剂苯甲酰胺处理经c-Ha-T24-ras活化癌基因转染得到的转化细胞系，处理4周后发现转化细胞系的某些细胞生物学特性发生了改变，呈现出正常细胞的某些特性。

This thesis includes five parts as follows.1. The backgrounds and some relative concepts of this work are briefly introduced. The photochemistry of benzamides and compounds with thiourea functional group is also concisely reviewed.2. Total of fourteen benzamides with different substituted groups have been synthesized and structurally characterized. Better photoreaction time for that kind of compounds at given concentrations is confirmed by tracking its'UV spectrum and GC chromatogram. A representative dibenzophenone photoproduct has been determined by X-ray crystallography. The mechanisms of photoreaction of benzamide have been proposed.3. Total of seven N-chloro(phenylmethylenebenzenamines with different substituted groups and sixty-one thiourea derivatives have been synthesized and structurally characterized.

论文的主要内容如下：1、简要介绍本论文工作的研究背景，并对苯甲酰胺和具有硫脲官能团类化合物的光化学研究进展进行简要的总结。2、合成与表征了14个具有不同取代基的苯甲酰胺类化合物，利用紫外光谱和气相色谱确定了此类化合物较佳光照时间，测定了一个具有代表性光解产物的单晶结构，提出了苯甲酰胺类化合物的光反应机理。3、合成与表征了7个带有不同取代基的氯代苯甲酰亚胺中间体及61个硫脲衍生物，测定了两个具有代表性化合物的单晶结构。

After treatment of benzamide which is an inhibitor of poly polymerase,β-galactosidase activity assays and PCR analysis were performed to test the deletion of LacZ gene and c-Ha-T24ras gene. The results showed that:(1)LacZ gene was deleted from both A13.4-NIH3T3 cells and B12.7-NIH3T3 cells, but neigher from A13.4-HeLa cells nor B12.7-HeLa cells. So it is possible that there is cell line specificity in gene deletion induced by BA.(2) In A13.4-NIH3T3 cells, LacZ gene and c-Ha-T24ras gene were completely deleted at the same time.(3) The transcription activity of exgenous DNA fragment may have same effect on its sensitivity to the deletion induced by BA.

用聚ADP核糖聚合酶的NAD位点抑制剂苯甲酰胺分别处理四种转化细胞后，检测细胞中整合的外源LacZ基因与c-Ha-T24ras基因的删除情况，结果如下：BA诱导的基因删除可发生于NIH3T3转化细胞系，但不能发生于HeLa转化细胞系；位于同一外源表达载体上的LacZ基因与c-Ha-T24ras基因的删除过程是同步的；外源整合DNA片段的转录强度可能直接影响其被BA诱导删除的敏感性。

The split between the two groups can hardly be papered over.

这两个团体间的分歧难以掩饰。

This approach not only encourages a greater number of responses, but minimizes the likelihood of stale groupthink.

这种做法不仅鼓励了更多的反应，而且减少跟风的可能性。