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In vitro time-killing studies, the combination of pei-amphotericin b and pei-fluconazole enhanced antifungal activity, but there was an antagonist for the combination of pei-polymyxin b.conclusionspei alone and in combination with amphotericin b and fluconazole displayed the high antifungal activity against candida albicans.

在体外致死研究实验中可以看到，pei-两性霉素b和pei-氟康唑结合物可以提高抑菌作用，但pei-多黏菌素b结合物却拮抗抑菌作用。结论 pei单独与联合使用均对白念珠菌产生很好的抗菌效果。

Caffeine (the agonist of RyR1) and ruthenium red (the antagonist of RyR1) had no effect on the E value either.

激动剂咖啡因，抑制剂钌红也不改变RyR1的E值。

By pretreatment with ruthenium red (RR, 100 1 μmol/L), an antagonist of vanilloid receptor subtype 1 (VR1), the above effects of CAP on carotid baroreflex were abolished.

2用香草酸受体亚型(vanilloid receptor subtype 1， VR1)阻断剂钌红(ruthenium red， 100 μmol/L)预处理后，CAP的上述反射效应即被阻断。

The concentration-response curve of GABA was shifted downward by hypotonic without any change of the threshold value.The values of two curves were very close(33.02μM and 29.41μM). Hypotonic decreased the maximal amplitude of IGABA by(31.38±2.13)%.③This inhibitory effect was reversed by ruthenium red, a nonselective TRPV4 receptor antagonist, and was increased by 4ɑ-PDD, a selectively TRPV4 receptor agonist.

低渗透压+GABA的量效曲线较单独的IGABA量效曲线明显下移，而两者的阈值和最大反应浓度基本不变，分别为10μM和1000μM；两条曲线的EC50值非常接近，分别为29.41μM和33.02μM；预加低渗透压后最大反应浓度时，IGABA的幅值减少了(31.38±2.13)%。

This inhibitory effect was increased by 4ɑ-PDD, a selective TRPV4 receptor agonist, and was reversed by ruthenium red, a nonselective TRPV4 receptor antagonist, suggesting that the inhibition is mediated via TRPV4 receptor.

4低渗透压对IATP的抑制作用可被TRPV4(transient receptor potential vanilloid 4)受体激动剂4ɑ-PDD(4ɑ-phorbol 12，13-didecanoate)增强，并可被TRPV4受体非特异性阻断剂钌红(ruthemium red， RR)阻断。

The excitatory response to intracarotid injection of capsaicin was significantly inhibited by pretreatment with the vanilloid receptor antagonist ruthenium red (200mmol, 0.1ml), The results indicate that capsaicin may activate the neurons of the brainstem nuclei involved in cardiovascular regulation through vanilloid receptors, but does not exert any effects on PAG and RN.

应用辣椒素受体阻断剂钌红(RR； 200mmol， 0.1 ml)，可明显抑制辣椒素的上述效应。以上结果提示，辣椒素可通过激活辣椒素受体，引起脑干内多个心血管活动相关核团的神经元兴奋，但对PAC和RN无影响。

Earlier study of this laboratory also showed that losartan, a selective antagonist of angiotensin Ⅱ type 1 receptor, alleviated BLM induced pulmonary fibrosis in rats.

我们实验室的前期研究表明Ang Ⅱ的一型受体AT1R的特异性拮抗剂氯沙坦能减轻BLM导致的大鼠肺纤维化。

RESULTS: We found that (1) tramadol, similar to the well-knownTRPV1 agonist, capsaicin, significantly increased [Ca2+] i ofTRPV1-CHO cells in a concentration-dependent fashion;(2) itseffect was reversibly prevented by the TRPV1 antagonist capsazepine;(3) repeated application of tramadol resulted in marked tachyphylaxis;and (4) tramadol did not modify [Ca2+] i in control CHO cells.

结果：我们发现以下结果：（1）曲马多和辣椒素这个熟知的辣椒素受体激动剂一样，呈浓度依赖性地显著增加 CHO 细胞 TRPV1内流钙离子；（2）该作用可以被 TRPV1拮抗剂 capsazepine 可逆性地阻止；（3）重复给予曲马多会造成显著的快速耐药性；（4）曲马多不修饰钙对照 CHO 细胞中的内流钙离子。

Methods: The effect of IL-1 and interleukin-1 receptor antagonist (IL -1ra) injected icv.on behavior and EEG of cortex and hippocampus were observed in rats with seizure induced by pentylenetetrazol.

采用记录脑电图同时观察行为的方法，观察IL-1β和IL-1受体拮抗剂(IL-1ra)侧脑室注射对戊四氮致痫大鼠行为和皮层、海马EEG的影响。

Rabeprazole belongs to a class of antisecretory compounds ( benzimidazole proton-pump inhibitors) that do not exhibit anticholinergic or histamine H2 -receptor antagonist properties, but suppress gastric acid secretion by inhibiting the gastric H +/K +-ATPase at the secretory surface of the gastric parietal cell.

雷贝拉唑属于抗分泌药物，苯并咪唑的替代品，质子泵抑制剂。不具有抗胆碱活性和组胺h2受体拮抗活性，但是能够胃壁细胞分泌表面的H +/K +-ATPase而抑制胃酸分泌。

The work of this paper is as follows: 1. Looking back the progressing history of the linear motor, introducing the features of the elevator driven by linear induction motor, radicating the topic of this paper "the digital frequency variable control of the elevator bi-side direct driven by linear induction motor". The research of this paper covers the conventional VVVF control, space vector based VVVF control, vector control and DTC.

本文主要开展了以下几个方面的工作： 1 回顾了直线电机发展历史，电机的驱动技术演变，特别是针对直线电机的驱动，简要介绍了直线感应电机驱动电梯的优点和不同结构类型，对传统的v／f控制，基于空间矢量法的v／f控制，矢量控制，和基于电压空间矢量的直接转矩控制进行了比较，确立了本课题的研究主题：直线感应电机双边直推式驱动电梯的全数字变频控制。

The article combines with the treatment of a superficial civil air defense work to introduce how the grouting method to improve the performance of the backfill soil.

文章从治理漂浮人防工事的角度提出了注浆技术在改善回填土性质方面的应用，并详细阐述了注浆技术的施工流程。